
Hello Bio/Ketanserin tartrate/HB1641/
市场价:
¥1150.50
美元价:
885.00
产品分类:
酸碱缓冲液
联系Q Q:
3392242852
电话号码:
4000-520-616
电子邮箱:
info@ebiomall.com
商品介绍
Productoverview
- NameKetanserintartrate
- ShortdescriptionSelective5-HT2receptorantagoNIST
- BIOLOGicaldescriptionSelective5-HT2SEROtoninreceptorantagonist.Showsdose-dependentα-1adrenoceptorinhibition.Usedtodifferentiatebetween5-HT1Dsubtypesbyshowingselectivityfor5-HT1Dα.Showsantihypertensive,antidepressantandanti-leishmaniasisactions.
- AlternativenamesR41468
- BiologicalactionAntagonist
- Purity>97%
- OurproductsinactionSubmitYourCitationNow
Properties
- Chemicalname3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3H]-quinazolinedionetartrate
- MolecularWeight545.52
- Chemicalstructure
- MolecularFormulaC22H22FN3O3.C4H6O6
- CASNumber83846-83-7
StoringandUsingYourProduct
- Storageinstructionsroomtemperature
- ImportantThisproductisforRESEARCHUSEONLYandisnotintendedfortherapeuticordiagnosticuse.Notforhumanorveterinaryuse.
ReferencesforKetanserintartrate
Antihypertensivepropertiesofketanserin(R41468).
VanhouttePMetal(1983)FedProc42(2):182-5.PubMedID:6295821DifferencesintheeffectsofketanserinandGR127935on5-HT-receptormediatedresponsesinrabbitsaphenousveinandguinea-pigjugularvein.
RazzaqueZetal(1995)EurJPharmacol283(1-3):199-206.PubMedID:7498311Ketanserin,anantidepressant,exertsitsantileishmanialactionviainhibitionof3-hydroxy-3-methylglutarylcoenzymeAreductase(HMGR)enzymeofLeishmaniadonovani.
SinghSetal(2014)ParasitolRes113(6):2161-8.PubMedID:24728519
品牌介绍
Hello Bio是由一群经验丰富的科学家和化学家们创立的充满活力的生物企业,总部位于英国布里斯托尔,在美国普林斯顿设有分公司,主旨在于提供质优价廉的生命科学研究工具,主要产品线为小分子化合物,如激动剂、拮抗剂、抑制剂等,部分产品价格甚至低至其他供应商的50%。热销产品线:酶抑制剂和激动剂ROCK inhibitor Y-27632, PKA inhibitor KT 5720 , adenylyl cyclase activator Forskolin, and novel GRK2/3 inhibitor Cmpd101等。 离子通道调节剂NMDA antagonist D-AP5, sodium channel blocker tetrodotoxin citrate, TRP antagonist capsazepine, and GABAA antagonist SR 95531 等。信号通路工具各种信号通路抑制剂、激动剂表观遗传学研究工具potent HDAC inhibitor Trichostatin A, DNA methyltransferase inhibitor 5-aza-2'-deoxycytidine,BET bromodomain inhibitor (+)-JQ1 and potent,selective GLP / G9a HMTase inhibitor BIX 01294 等受体配体novel selective GRK2/3 inhibitor, NMDA antagonist D-AP5, Group I mGlu agonist (S)-3,5-DHPG, and GABAA antagonist SR 95531.等干细胞调节剂ROCK inhibitor Y-27632, SB 431542 DAPT.
联络我们