
你好Bio/AZM 475271/HB1322/50mg
商品编号:
HB1322-50mg
品牌:
hellobio
市场价:
¥8970.00
美元价:
6900.00
产品分类:
酸碱缓冲液
联系Q Q:
3392242852
电话号码:
4000-520-616
电子邮箱:
info@ebiomall.com
商品介绍
Productoverview
- NameAZM475271
- ShortdescriptionSrctyrosinekinaseinhibitor
- BIOLOGicaldescriptionSrctyrosinekinaseinhibitor.Showsanti-proliferative,apoptotic,anti-angiogenic,anti-lymphangiogenicandantimetastaticactionsagainstcancer.
- BiologicalactionInhibitor
- Purity>99%
- OurproductsinactionSubmitYourCitationNow
Properties
- ChemicalnameN-(2-Chloro-5-methoxyphenyl)-6-methoxy
- MolecularWeight442.94
- MolecularFormulaC23H27ClN4O3
- CASNumber476159-98-5
StoringandUsingYourProduct
- Storageinstructionsroomtemperature
- SolubilityoverviewsolubleinDMSO(100mM)
- ImportantThisproductisforRESEARCHUSEONLYandisnotintendedfortherapeuticordiagnosticuse.Notforhumanorveterinaryuse.
ReferencesforAZM475271
InhibitionofSRCtyrosinekinaseastreatmentforhumanpancreaticcancergrowingorthotopicallyinnudemice.
YezhelyevMVetal(2004)ClinCancerRes10(23):8028-36.PubMedID:15585638EffectofSrckinaseinhibitiononmetastasisandtumorangiogenesisinhumanpancreaticcancer.
IschenkoIetal(2007)Angiogenesis10(3):167-82.PubMedID:17486419Srctyrosinekinaseinhibitionsuppresseslymphangiogenesisinvitroandinvivo.
IschenkoIetal(2010)CurrCancerDrugTargets10(5):546-53.PubMedID:20370688
品牌介绍
Hello Bio是由一群经验丰富的科学家和化学家们创立的充满活力的生物企业,总部位于英国布里斯托尔,在美国普林斯顿设有分公司,主旨在于提供质优价廉的生命科学研究工具,主要产品线为小分子化合物,如激动剂、拮抗剂、抑制剂等,部分产品价格甚至低至其他供应商的50%。热销产品线:酶抑制剂和激动剂ROCK inhibitor Y-27632, PKA inhibitor KT 5720 , adenylyl cyclase activator Forskolin, and novel GRK2/3 inhibitor Cmpd101等。 离子通道调节剂NMDA antagonist D-AP5, sodium channel blocker tetrodotoxin citrate, TRP antagonist capsazepine, and GABAA antagonist SR 95531 等。信号通路工具各种信号通路抑制剂、激动剂表观遗传学研究工具potent HDAC inhibitor Trichostatin A, DNA methyltransferase inhibitor 5-aza-2'-deoxycytidine,BET bromodomain inhibitor (+)-JQ1 and potent,selective GLP / G9a HMTase inhibitor BIX 01294 等受体配体novel selective GRK2/3 inhibitor, NMDA antagonist D-AP5, Group I mGlu agonist (S)-3,5-DHPG, and GABAA antagonist SR 95531.等干细胞调节剂ROCK inhibitor Y-27632, SB 431542 DAPT.
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